Guillon, R.
Publications
P212
Eur. J. Med. Chem. 2020, 189, 112082.
New Azole Antifungals with a Fused Triazinone Scaffold.
doi: 10.1016/j.ejmech.2020.112082
P116
Tetrahedron, 2013, 69, 3182-3191.
Novel synthesis of angular thiazolo[5,4-f] and [4,5-h]quinazolines, preparation of their linear thiazolo[4,5-g] and [5,4-g]quinazoline analogs.
P114
ACS Med. Chem. Lett., 2013, 4, 288-292.
Discovery of a novel broad-spectrum antifungal agent, derived from albaconazole.
P96
ChemMedChem, 2011, 6, 1806-1815.
Design, synthesis and biological evaluation of 1-[(biarylmethyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as potent antifungal agents: new insights into structure-activity relationships.
P91
ChemMedChem, 2011, 6, 816-825.
Design, synthesis and in vitro antifungal activity of 1-[(4-substituted benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
P87
J. Enzym. Inhib. Med. Chem., 2011, 26(2), 261-269.
Synthesis and in vitro antifungal evaluation of 2-(2,4-difluorophenyl)-1-[(1H-indol-3-ylmethyl)methylamino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
P79
Bioorg. Med. Chem. Lett., 2009, 19(20), 5833-5836.
Design of new antifungal agents: synthesis and evaluation of 1-[(1H-indol-5-ylmethyl)amino]-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
P74
Bioorg. Med. Chem. Lett., 2009, 19(2), 301-304
Synthesis and structure-activity relationships of 2-phenyl-1-[(pyridinyl- and piperidinylmethyl)amino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents.
Autres publications scientifiques
Brevets
B17.
Novel fused pyrimidone and triazinone derivatives containing bridged nitrogen, their process of preparation and their therapeutic uses as antifungal and/or antiparasitic agents.
PCT WO 2017/021178 A1, 9 février 2017.
Thèse
T25.
Conception, synthèse et évaluation pharmacologique de nouveaux azolés à activité antifongique.
Nantes, date de soutenance : 1er octobre 2010.