Publications
P302
Inorg. Chem., 2025, 64, 16192-16203.
Synthesis and Biological Evaluation of Itraconazole Derivatives: Design in an Old Scaffold.
https://doi.org/10.1021/acs.inorgchem.5c02730
P300
RSC Med. Chem. 2025, 16, 3746–3763.
Pharmacophore-guided optimization of the hit compound CTN1122 in the design of promising imidazo[1,2-a]pyrazine derivatives targeting the casein kinase 1 for antileishmanial therapy
https://doi.org/10.1039/D5MD00257E
P290
ChemMedChem. 2025, 20, e202400862.
Investigating the C2 modulation of the imidazo[1,2-a]pyrazine-based hit compound CTN1122: synthesis, in vitro antileishmanial activity, cytotoxicity and casein kinase 1 inhibition.
https://doi.org/10.1002/cmdc.202400862
P280
Chem. Biodiversity 2024, e202300563
Chemical Composition, Antifungal, Antioxidant, and Hemolytic Activities of Morrocan Thymus capitatus Essential Oil.
https://doi.org/10.1002/cbdv.202300563
P270
J. Fungi 2023, 9, 430.
The mortality attributable to candidemia in C. auris is higher than that in other Candida species: Myth or reality?
https://doi.org/10.3390/jof9040430
P269
Nat. Prod. Res. 2023
Phytochemical, antileishmanial, antifungal and cytotoxic profiles of Thymelaea tartonraira (L.) All. extracts.
https://doi.org/10.1080/14786419.2023.2252153
P251
Microorganisms. 2022, 10, 938.
Prototheca infections and ecology from a One Health perspective.
https://doi.org/10.3390/microorganisms10050938
P234
Med. Chem. Res. 2021, 30, 152-162.
Antimicrobial and anti-leishmanial activities of extracts and some constituents from the leaves of Solanum chrysotrichum Schldl.
doi: 10.1007/s00044-020-02648-8
P231
Eur. J. Med. Chem. 2021, 210, 112956.
In vitro identification of imidazo[1,2-a]pyrazine-based antileishmanial agents and evaluation of L. major casein kinase 1 inhibition.
doi: 10.1016/j.ejmech.2020.112956
P212
Eur. J. Med. Chem. 2020, 189, 112082.
New Azole Antifungals with a Fused Triazinone Scaffold.
doi: 10.1016/j.ejmech.2020.112082
P208
J. Enzym. Inhib. Med. Chem. 2020, 35, 398-403.
Biological exploration of a novel 1,2,4-triazole-indole hybrid molecule as antifungal agent.
doi: 10.1080/14756366.2019.1705292
P136
Eur. J. Med. Chem. 2015, 103, 381-395.
Synthesis, antileishmanial activity and cytotoxicity of 2,3-diaryl- and 2,3,8-trisubstituted imidazo[1,2-a]pyrazines.
doi: 10.1016/j.ejmech.2015.09.002
P114
ACS Med. Chem. Lett., 2013, 4, 288-292.
Discovery of a novel broad-spectrum antifungal agent, derived from albaconazole.
P108
Eur. J. Med. Chem., 2012, 58, 543-556.
Synthesis and biological evaluation of 2,3-diarylimidazo[1,2-a]pyridines as antileishmanial agents.
P96
ChemMedChem, 2011, 6, 1806-1815.
Design, synthesis and biological evaluation of 1-[(biarylmethyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as potent antifungal agents: new insights into structure-activity relationships.
P91
ChemMedChem, 2011, 6, 816-825.
Design, synthesis and in vitro antifungal activity of 1-[(4-substituted benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
P87
J. Enzym. Inhib. Med. Chem., 2011, 26(2), 261-269.
Synthesis and in vitro antifungal evaluation of 2-(2,4-difluorophenyl)-1-[(1H-indol-3-ylmethyl)methylamino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
P79
Bioorg. Med. Chem. Lett., 2009, 19(20), 5833-5836.
Design of new antifungal agents: synthesis and evaluation of 1-[(1H-indol-5-ylmethyl)amino]-2-phenyl-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
P77
J. Enz. Inh. Med. Chem., 2009, 24(5), 1067-1075.
Design, synthesis and evaluation of 3-(imidazol-1-ylmethyl)indoles as antileishmanial agents. Part II.
P74
Bioorg. Med. Chem. Lett., 2009, 19(2), 301-304
Synthesis and structure-activity relationships of 2-phenyl-1-[(pyridinyl- and piperidinylmethyl)amino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as antifungal agents.
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