Robert, J-M. | IICIMED

Robert, J-M.

Publications

P88

Cell Death and Differentiation, 2011, 18(3), 528-537.

Prostaglandins antagonistically control Bax activation during apoptosis.


P68

Bioorg. Med. Chem. 2008, 16(9), 4932-4953.

Synthesis of 3,5-bis(2-indolyl)pyridine and 3-[(2-indolyl)-5-phenyl]pyridine derivatives as CDK inhibitors and cytotoxic agents.


P64

J. Enz. Inh. Med. Chem. 2008, 23(5), 659-667.

Synthesis and immunosuppressive activity evaluation of substituted N-imidazolidin-2-ones and N-tetrahydropyrimidin-2(1H)-ones.


P59

Eur. J. Med. Chem., 2008, 43(7), 1469-1477.

Novel 9-oxo-thiazolo[5,4-f]quinazoline-2-carbonitrile derivatives as dual cyclin-dependent kinase 1 (CDK1) / glycogen synthase kinase-3 (GSK-3) inhibitors: synthesis, biological evaluation and molecular modeling studies.


P53

Bioorg. Med. Chem. Lett. 2006, 16, 3419-3423.

Thiazolo[5,4-f]quinazolin-9-ones, inhibitors of glycogen synthase kinase-3.


P45

J. Enz. Inh. Med. Chem. 2005, 20, 581-585.

Three-Dimensional Model of Cytochrome P450 Human Aromatase.


P36

Tetrahedron 2004, 60, 6079-6083.

Synthesis of 1-benzyl-8,9-dihydroimidazo[4,5-c]pyrrolo[3,2-g]quinolin-4(5H)-one via palladium-catalyzed intramolecular arylation.


P33

Eur. J. Med. Chem. 2003, 38, 711-718.

Synthesis and antileismanial activity of new imidazolidin-2-one derivatives.


P16

J. Enz. Inh. Med. Chem. 2002, 17, 443-447.

 Inhibition of protein kinase C by new antileishmanial imidazolidin-2-one compounds.


P15

Parasite 2002, 9, 367-370. 

In vitro and in vivo antileishmanial activity of 2-amino-4,6-dimethylpyridine derivatives against Leishmania mexicana.


P14

Eur. J. Pharmacol. 2001, 431, 103-110.

Effects of tumour necrosis factor-a synthesis inhibitors on rat trinitrobenzene sulphonic acid-induced chronic colitis.


P12

 Eur. J. Med. Chem. 2001, 36, 639-649.

New antiinflammatory N-pyridinyl(alkyl)phtalimides acting as tumor necrosis factor-a production inhibitors. 


P9

J. Pharm. Pharmacol. 2001, 53, 417-423.

Synthesis of N-pyridinyl(methyl)-1,2-dihydro-4-hydroxy-2-oxoquinoline-3-carbo-xamides and analogues and their anti-inflammatory activity in mice and rats.


P7

Arzneim.-Forsch./Drug Res. 2000, 50 (I), 479-484.

Synthesis and antileishmanial activity of new 1-(pyridin-2-yl)imidazolidin-2-ones derived from 2-amino-4,6-dimethylpyridine.


P6

Pharm. Pharmacol. Commun. 1999, 5, 233-238.

N-Pyridinyl(alkyl)polyhalogenobenzamides acting as TNF-a production inhibitors. 


P5

Acta. Parasitologica 1999, 44, 156-159.

Activity of N-lutidinylarylcarboxamides against Leishmania donovani and L. braziliensis. 


P3

Bioorg. Med. Chem. Lett. 1999, 9, 333-336.

New selective nonsteroidal aromatase inhibitors: synthesis and inhibitory activity of 2, 3 or 5-(a-azolylbenzyl)-1H-indoles.


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