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Int. J. Mol. Sci. 2021, 22, 7763.

Exosomes as New Biomarkers and Drug Delivery Tools for the Prevention and Treatment of Various Diseases: Current Perspectives.

Liu, Q. | Li, S. | Dupuy, A. | Mai, H.l. | Sailliet, N. | Logé, C. | Robert, J.-M.H. | Brouard, S.

doi: 10.3390/ijms22157763

P240

Molecules 2021, 26, 6572.

Dibenzofuran derivatives inspired from cercosporamide as dual inhibitors of Pim and CLK1 kinases.

Dao, V. H. | Ourliac-Garnier, I. | Logé, C. | McCarthy, F. O. | Bach, S. | da Silva, T. G. | Denevault-Sabourin, C. | Thiéfaine, J. | Baratte, B. | Robert, T. | Gouilleux, F. | Brachet-Botineau, M. | Bazin, M.-A. | Marchand, P.

doi: 10.3390/molecules26216572

P239

Chem. Biol. Interact. 2021, 347, 109597.

Synthesis, anticancer activity and mechanism of action of new phthalimido-1,3-thiazole derivatives.

Rodrigues Oliveira, A. | Alves dos Santos, F. | de Lima Ferreira, L. P. | da Rocha Pitta, M. G. | de Oliveira Silva, M. V. | de Oliveira Cardoso, M. V. | Ferreira Pinto, A. | Marchand, P. | Barreto de Melo Rêgo, M. J. | Lima Leite, A. C.

doi: 10.1016/j.cbi.2021.109597

P238

Med. Chem. Lett. 2021, 47,  128196.

Anti-protozoal and anti-fungal evaluation of 3,5-disubstituted 1,2-dioxolanes. Bioorg.

Pinet, A. | Cojean, S. | Nguyen, L. T. | Vásquez-Ocmín, P. | Maciuk, A. | Loiseau, P. M. | Le Pape, P. | Figadère, B. | Ferrié, L.

doi: 10.1016/j.bmcl.2021.128196

P237

Phytochem. Lett. 2021, 43, 212-218.

New cyclolignans of Larrea tridentata and their antibacterial and cytotoxic activities.

Núñez-Mojica, G. | Vázquez-Ramírez, A. L. | García, A. | Rivas-Galindo, V. M. | Garza-González, E. | Cuevas González-Bravo, G. E. | Toscano, R. A. | Moo-Puc, R. E. | Villanueva-Toledo, J. R. | Marchand, P. | Camacho-Corona, M. R.

doi: 10.1016/j.phytol.2021.04.013

P236

J. Glob. Antimicrob. Resist. 2021, 25, 171-180.

Characterisation of the antifungal effects of a plant-based compound, CIN-102, on the main septal filamentous fungi involved in human pathology.

D'Agostino, M. | Tesse, N. | Lavergne, R.-A. | Le Pape, P. | Bouchara, J.-P. | Frippiat, J.-P. | Machouart, M. | Debourgogne, A.

doi: 10.1016/j.jgar.2021.03.017

P235

Atlas of Science. 2021.

Allosteric degraders of EGFR leading to cancer cell detachment-promoted death.

Iradyan, M. | Iradyan, N. | Sakanyan, V.

P234

Med. Chem. Res. 2021, 30, 152-162.

Antimicrobial and anti-leishmanial activities of extracts and some constituents from the leaves of Solanum chrysotrichum Schldl.

Núñez-Mojica, G. | Rivas-Galindo, V. M. | Garza-González, E. | Miranda, L. D. | Romo-Pérez, A. | Pagniez, F. | Picot, C. | Le Pape, P. | Bazin, M.-A. | Marchand, P. | Camacho-Corona, M. R.

doi: 10.1007/s00044-020-02648-8

P233

Drug Discov. Today. 2021, 26, 56-68.

Tetraspanins: useful multifunction proteins for the possible design and development of small-molecule therapeutic tools.

Robert, J.-M. H. | Amoussou, N. G. | Le Mai, H. | Logé, C. | Brouard, S.

doi: 10.1016/j.drudis.2020.10.022

P232

 Chem. Biol. Interact. 2021, 333, 109316. 

Streptomyces hygroscopicus UFPEDA 3370: a valuable source of the potent cytotoxic agent nigericin and its evaluation against human colorectal cancer cells.

Rodini Garcia Princival, I. M. | Princival, J. L. | Dias da Silva, E. | de Arruda Lima, S. M. | Carvalho Carregosa, J. | Wisniewski Jr, A. | Oliveira de Lucena, C. C. | Halwass, F. | Alves Franca, J. A. | Gomes Rebello Ferreira, L. F. | Zaldini Hernandes, M. | Alcântara Saraiva, K. L. | Alves Peixoto, C. | Baratte, B. | Robert, T. | Bach, S. | Correia Gomes, D. | Guedes Paiva, P. M. | Marchand, P. | do Desterro Rodrigues, M. | Gonçalves da Silva, T.

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P231

Eur. J. Med. Chem. 2021, 210, 112956.

In vitro identification of imidazo[1,2-a]pyrazine-based antileishmanial agents and evaluation of L. major casein kinase 1 inhibition.

Bazin, M.-A. | Cojean, S. | Pagniez, F. | Bernadat, G. | Cavé, C. | Ourliac-Garnier, I. | Nourrisson, M.-R. | Morgado, C. | Picot, C. | Leclercq, O. | Baratte, B. | Robert, T. | Späth, G.F. | Rachidi, N. | Bach, S. | Loiseau, P.M. | Le Pape, P. | Marchand, P.

doi: 10.1016/j.ejmech.2020.112956