Robert, T. | IICIMED

Robert, T.

Publications

P300

RSC Med. Chem. 2025, 16, 3746–3763. 

 Pharmacophore-guided optimization of the hit compound CTN1122 in the design of promising imidazo[1,2-a]pyrazine derivatives targeting the casein kinase 1 for antileishmanial therapy


https://doi.org/10.1039/D5MD00257E

P290

ChemMedChem. 2025, 20, e202400862.

Investigating the C2 modulation of the imidazo[1,2-a]pyrazine-based hit compound CTN1122: synthesis, in vitro antileishmanial activity, cytotoxicity and casein kinase 1 inhibition.


https://doi.org/10.1002/cmdc.202400862

P244

Letter to the Editor, Quim. Nova 2022, 45, 1-3.

The Franco-Brazilian Network on Natural Products (FB2NP): a new network promoting cooperation and exchanges in natural products research. 


https://doi.org/10.21577/0100-4042.20170847

P240

Molecules 2021, 26, 6572.

Dibenzofuran derivatives inspired from cercosporamide as dual inhibitors of Pim and CLK1 kinases.


doi: 10.3390/molecules26216572

P231

Eur. J. Med. Chem. 2021, 210, 112956.

In vitro identification of imidazo[1,2-a]pyrazine-based antileishmanial agents and evaluation of L. major casein kinase 1 inhibition.


doi: 10.1016/j.ejmech.2020.112956

P178

Eur. J. Med. Chem. 2018, 154, 101-109.

Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors.


doi: 10.1016/j.ejmech.2018.04.056

P177

Bioorg. Med. Chem. 2018, 26, 4209-4224.

Synthesis and anticancer activity of novel bisindolylhydroxymaleimide derivatives with potent GSK-3 kinase inhibition.


doi: 10.1016/j.bmc.2018.07.012.

P102

Med. Mycol., 2012, 50(6), 594-600. 

Phaeohyphomycosis due to Alternaria infectoria: a single-center experience with utility of PCR for diagnosis and species identification.


Autres publications scientifiques

PS36

Pharmaceuticals 2025, 18, 837.

New insights into the anticancer effects and toxicogenomic safety of two β-Lapachone derivatives.


https://doi.org/10.3390/ph18060837

PS22

Molbank, 2023 

Potassium 6-oxo-7,13,16,22-tetraazatetracyclo[12.6.2.18,12.017,21]tricosa-1(20),8(23), 9,11,14,16,18,21-octaen-2-yne-15-carboxylate.


https://doi.org/10.3390/M1735

PS01

Molecules. 2021, 26,867

New quinoxaline derivatives as dual Pim-1/2 inhibitors: design, synthesis and biological evaluation.


https://doi.org/10.3390/molecules26040867

Brevets

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