Loidreau, Y. | IICIMED

Loidreau, Y.

Publications

P222

Pharmaceuticals. 2020, 13, 202.

Microwave-assisted synthesis of potential bioactive benzo-, pyrido- or pyrazino-thieno[3,2-d]pyrimidin-4-amine analogs of MPC-6827.


doi: 10.3390/ph13090202

P219

Pharmaceuticals 2020, 13, 89.

Exploring kinase inhibition properties of 9H-pyrimido[5,4-b]- and [4,5-b]indol-4-amine derivatives.


doi: 10.3390/ph13050089

P139

Eur. J. Med. Chem. 2015, 92, 124-134.

Synthesis and molecular modelling studies of 8-arylpyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-amines as multitarget Ser/Thr kinases inhibitors.


doi: 10.1016/j.ejmech.2014.12.038

P122

Bioorg. Med. Chem. Lett. 2013, 23, 6784-6788.

Synthesis of novel 7-substituted pyrido[2',3':4,5]furo[3,2-d]pyrimidin-4-amines and their N-aryl analogues and evaluation of their inhibitory activity against Ser/Thr Kinases.


P113

Eur. J. Med. Chem. 2013, 59, 283-295.

Synthesis and biological evaluation of N-aryl-7-methoxybenzo[b]furo[3,2-d]pyrimidin-4-amines and their N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amine analogues as dual inhibitors of CLK1 and DYRK1A kinases.


P112

J. Het. Chem., 2013, 50, 1187-1197.

Efficient new synthesis of N-arylbenzo[b]furo[3,2-d]pyrimidin-4-amines and their benzo[b]thieno[3,2-d]pyrimidin-4-amine analogues via a microwave-assisted Dimroth rearrangement.


PXXX

Org. Biomol. Chem. 2012, 10, 4916-4925

Study of N(1)-alkylation of indoles from the reaction of 2(or 3)-aminoindole-3-(or 2)carbonitriles with DMF-dialkylacetals


https://doi.org/10.1039/C2OB25747E

P107

Eur. J. Med. Chem., 2012, 58, 171-183.

Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors.


P100

Tetrahedron Lett., 2012, 53, 944-947. 

First synthesis of 4-aminopyrido[2',3':4,5]furo[3,2-d]pyrimidines.


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